Kinase Inhibitor Profiling: The best value services for kinase inhibitor profiling

Experience the first and only kinase inhibitor profiling service that gives you precise Kd values for your compounds on a full human kinome scale. Powered by our proprietary DIANA technology, we provide:


  • Unbeatable market pricing
  • Reliable quantitative potency insights (Kd values)
  • Exceptional customization and dedicated support
  • Fast and efficient turnaround


Download the complete DB Kinase Panel assay list here!


Download the full DIANA Kinase Inhibitor Profiling booklet here!

Services

Meet your highest standards with our proprietary Kinase Panels!

DB Kinase Panel™ is our flagship profiling package, covering over 170 kinases across the entire human kinome. Powered by proprietary DIANA technology, each run delivers true binding constants (Kd) for every kinase making DB Kinase Panel™ the only tool on the market for quantitative potency determination at full kinome scale.

The DB MiniKinase Panel™ is a precision-engineered set of 48 assays designed to represent the entire human kinome. By leveraging a proprietary optimization algorithm and inhibition "fingerprints" from over 257 kinases, this panel maximizes coverage while minimizing your screening footprint. Profile smarter with the industry's most efficient representative set.

We are continuously expanding the portfolio of assays in our kinase panel. We started with a set of assays that together provide a representative coverage of the entire human kinome. Currently, we are focusing on completing smaller, coherent groups of assays that can function as focused subpanels of our flagship product, the DB Kinase Panel™, gathered under our DB Focused Panel™ brand.

DIANA CDK panel is an advanced kinase inhibitor selectivity profiling tool which comprise 24 different CDK/cyclin complexes. Using proprietary DIANA technology it delivers quantitative affinity measurements (Kd) from single measurement.

DIANA CK1 panel is an advanced CK1 (casein kinase 1) inhibitor selectivity profiling tool which comprise 7 different CK1s. Using proprietary DIANA technology it delivers quantitative affinity measurements (Kd) from single measurement.

DIANA TK panel is an advanced tyrosine kinase inhibitor selectivity profiling tool which comprise 69 different TKs. Using proprietary DIANA technology it delivers quantitative affinity measurements (Kd) from single measurement.

Pricing of DIANA Kinase Inhibitor Profiling Services

Product Name

No. Kinases

Cpds

Price (EUR)

Price per kinase (EUR)

Turnaround Time**

Result

DB Kinase Panel

+170†

1

2500

15

14 business days

Dissociation constant (Kd)

DB MiniKinase Panel

48

2

1440***

20

7 business days

Dissociation constant (Kd)

DIANA TK Panel

70

1

1360

20

7 business days

Dissociation constant (Kd)

DIANA CDK Panel

24

1

480

20

7 business days

Dissociation constant (Kd)

DIANA CK1 Panel

7

1

140*

20

7 business days

Dissociation constant (Kd)

Custom selection

1

1

25*

25

7 business days

Dissociation constant (Kd)

*Minimal Order Quantity for Custom Selection service is 500 EUR.

**Counts from the day compounds are delivered to our testing facility. For complex orders the turnaround time can be extended to 14 business days.

***DB MiniKinase Panel can be ordered also for 1 cpds for 960 EUR.

†The list of kinases is constantly growing. For the most recent info, download the current list of kinases.


All prices exclude VAT.

Service without compromises

DIANA Assay: Accelerate Your Project and Get Quantitative Potency Data from the Start!

Get more for your price


Quantitative potency data for the price of relative potency data

Rapid turnaround time


7 business days for standard and 14 business days for complex services

Flexible customization


You can assemble your own kinase panel for comparable price as our focused panels

Whole kinome coverage


Our kinase assay portfolio representatively covers all kinase families within human kinome

“The services provided by DIANA Biotech in the area of discovery and profiling of kinase inhibitors have been seminal for rapid progression of several research projects in our group. Specifically, we have used the DIANA platform for HTS campaigns focused on two underexplored protein kinases (which delivered high-quality hits), and activity/selectivity profiling in several other projects. The data quality was consistently high and the price-performance ratio very favorable, with the promptly responding DIANA team providing top-class support. I can therefore highly recommend DIANA Biotech services in the area of protein kinase research.”

Kamil Paruch, PhD

Associate Professor at Masaryk's University

"After several years of regularly using Eurofins Scientific for kinase profiling, we recently decided to try DIANA Biotechnologies, a new Czech biotech initiative originating from the Czech Academy of Sciences. They offer comparable kinase screening services at a significantly lower cost, so we decided to give them a chance. I must say that the communication was excellent: our specific experimental needs were clearly understood, and the entire process was transparent from start to finish. The results were delivered within three weeks, and the DIANA team even provided additional support during data interpretation and manuscript preparation. Overall, our experience was highly positive, and we can confidently recommend DIANA Biotechnologies as a reliable and innovative partner for kinase screening studies."

Lukáš Górecki, PhD

Biomedical Research Centre, University Hospital Hradec Králové

Download all the materials!

Document name

Download

DB Kinase Panel™: List of kinases

Download

DB Inhibitor Profiling: Leaflet

Download

Technology Intro

What is DIANA Assay?

DIANA is a solid-phase competitive binding assay that uniquely combines small molecule-based DIANA probes with the strengths of ELISA and qPCR, delivering robust quantitative potency data with an exceptionally broad dynamic range. This allows researchers to obtain precise binding affinity constants (Kd) from the start of their projects at a cost comparable to conventional methods that only provide relative inhibition.

DIANA Assay

Competitive Binding Assay

DIANA assay measures potency of tested compound as function of its competition with DIANA probe. The assay delivers true binding constants (Kd) of test compound.

DIANA Assay

qPCR Readout

The amount of displaced DIANA probe is quantitatively determined by qPCR. qPCR readout ensures high dynamic range and enables calculation of Kd from a single measurement.

DIANA Assay

Superior to KINOMEscan

Similar assay setup yields highly comparable results between the methods. Usage of recombinant kinases instead of phage constructs ensures easier kinase quality control and consistency of results.

Consultation

Contact us to schedule complimentary consultation!

Not sure what you precisely need? Are you seeking an advice to your problems? Feel free to contact us to schedule consultation with our specialist directly.

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